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Inhibition of [3H]kainate binding to Ionotropic glutamate receptor kainate of central nervous system
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Percent inhibition against Kainate receptor at a compound concentration of 1 uM
Assay data:1 Active, 1 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibitory activity against kainic acid receptor using [3H]-kainic acid as radioligand
The compound was tested for binding affinity against Kainate binding site using [3H]kainate as radioligand; Not tested
SummaryRelated BioAssays by Target
The compound was tested for binding affinity against Kainate binding site using [3H]kainate as radioligand.
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
The compound was tested for binding affinity against Kainate binding site using [3H]kainate as radioligand
Assay data:8 Active, 1 Activity ≤ 1 µM, 8 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Ability to displace [3H]kainate from kainate receptor
Assay data:9 Active, 3 Activity ≤ 1 µM, 10 Tested
Inhibition of binding of [3H]kainate to kainate at 10 uM compound concentration
Compound has been evaluated for its binding affinity towards kainate by displacing the radioligand [3H]kainate
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibitory activity against Ionotropic glutamate receptor kainate using [3H]- Kainate at 10e5 (M)
Percentage binding to kainate receptor at 10 uM
Compound was tested for binding affinity against Ionotropic glutamate receptor kainate using [3H]kainate as a radioligand.; Not tested
Assay data:4 Tested
Compound was tested for binding affinity against Ionotropic glutamate receptor kainate using [3H]kainate as a radioligand.
Assay data:6 Active, 1 Activity ≤ 1 µM, 6 Tested
Tested for the affinity for the Ionotropic glutamate receptor kainate using [3H]kainate as radioligand
Assay data:2 Active, 6 Tested
In vitro binding affinity against Ionotropic glutamate receptor kainate (kainic acid) using [3H]KAIN as radioligand
Assay data:1 Active, 10 Tested
Binding affinity against Ionotropic glutamate receptor kainate using [3H]-Kainic acid as a radioligand; NT = Not tested
Binding affinity against Ionotropic glutamate receptor kainate using [3H]-Kainic acid as a radioligand
Compound was evaluated to potentiate response to Ionotropic glutamate receptor kainate
siRNA Circadian Assay
Assay data:527 Active, 33364 Tested
SummaryPubMed CitationRelated BioAssays by Depositor
Druggable Genome siRNA Screen for Enhancers of Camptothecin in MDA-MB-231 Breast Cancer Cells
Assay data:167 Active, 26449 Tested
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