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Inhibitory activity against Ionotropic glutamate receptor kainate using [3H]- Kainate at 10e5 (M)
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
The compound was tested for binding affinity against Kainate binding site using [3H]kainate as radioligand.
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
The compound was tested for binding affinity against Kainate binding site using [3H]kainate as radioligand
Assay data:8 Active, 1 Activity ≤ 1 µM, 8 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Ability to displace [3H]kainate from kainate receptor
Assay data:9 Active, 3 Activity ≤ 1 µM, 10 Tested
Inhibition of binding of [3H]kainate to kainate at 10 uM compound concentration
Compound has been evaluated for its binding affinity towards kainate by displacing the radioligand [3H]kainate
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Binding affinity towards cloned human Kai-2 subunit stably expressed in cultured HEK293 cells using [3]H-kainate as radioligand
Assay data:1 Active, 8 Tested
Binding affinity towards Kai-2 using [3]H-kainate as the radioligand
Assay data:1 Active, 3 Tested
Compound was tested for binding affinity against Ionotropic glutamate receptor kainate (KA2) in HK293 cells
Ability to bind to Ionotropic glutamate receptor kainate (kainate 2) was evaluated.
Assay data:2 Active, 2 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]kainate from human Ionotropic glutamate receptor ionotropic kainate 1 expressed in HEK293 cells
Assay data:13 Active, 1 Activity ≤ 1 nM, 9 Activity ≤ 1 µM, 14 Tested
Electrophysiological data on Xenopus oocytes, expressing homomeric kainate receptor (GluR5)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Electrophysiological data on Xenopus oocytes, expressing homomeric Ionotropic glutamate receptor ionotropic kainate 1 (GluR5)
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
The compound was tested for binding affinity against Kainate binding site using [3H]kainate as radioligand; Not tested
SummaryRelated BioAssays by Target
Inhibition of [3H]kainate binding to Ionotropic glutamate receptor kainate of central nervous system
Compound was tested for binding affinity against Ionotropic glutamate receptor kainate using [3H]kainate as a radioligand.; Not tested
Assay data:4 Tested
Compound was tested for binding affinity against Ionotropic glutamate receptor kainate using [3H]kainate as a radioligand.
Assay data:6 Active, 1 Activity ≤ 1 µM, 6 Tested
Tested for the affinity for the Ionotropic glutamate receptor kainate using [3H]kainate as radioligand
Assay data:2 Active, 6 Tested
In vitro binding affinity against Ionotropic glutamate receptor kainate (kainic acid) using [3H]KAIN as radioligand
Assay data:1 Active, 10 Tested
Binding affinity against Ionotropic glutamate receptor kainate using [3H]-Kainic acid as a radioligand; NT = Not tested
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