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Activity at human B2 receptor transfected in CHO cells assessed as ability to antagonize BK-induced inositol-phosphate accumulation
Assay data:18 Active, 1 Activity ≤ 1 nM, 18 Activity ≤ 1 µM, 21 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of radiolabeled NPC 567 from human bradykinin B2 receptor
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to human bradykinin B2 receptor at 10 uM relative to control
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of human bradykinin B2 receptor at 10 uM
Inhibition of human bradykinin B2 receptor at 1 uM
Assay data:3 Tested
Inhibition of human bradykinin B2 receptor
Binding affinity at bradykinin B2 receptor at 1 uM
Inhibition of bradykinin B2 receptor at 1 uM
Displacement of [3H]bradykinin from human bradykinin B2 receptor expressed in CHO cells
Antagonist potency at human bradykinin B2 receptor assessed as effect on inositol monophosphate accumulation in CHOdhfr- cells
Assay data:34 Active, 14 Activity ≤ 1 nM, 34 Activity ≤ 1 µM, 34 Tested
Displacement of [3H]BK from human bradykinin B2 receptor transfected in CHO cells
Assay data:34 Active, 32 Activity ≤ 1 nM, 34 Activity ≤ 1 µM, 34 Tested
Displacement of [3H]bradykinin from human bradykinin B2 receptor expressed in CHO-K1 cells
Assay data:12 Tested
Assay data:9 Tested
Inhibition of human B2 receptor at 10 uM
Inhibition of B2 receptor at 1 uM
Binding affinity to CCK1 receptor
Assay data:3 Active, 3 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Displacement of [3H]BK from human B2 receptor transfected in CHO cells
Assay data:56 Active, 10 Activity ≤ 1 nM, 50 Activity ≤ 1 µM, 56 Tested
Antagonist activity against bradykinin B2 receptor
Assay data:2 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 3 Tested
Binding affinity to human bradykinin B2 receptor transfected in CHO cells
Assay data:3 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 3 Tested
Binding affinity to bradykinin B2 receptor at 10 uM
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