Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Adenosine A1 Eurofins Panlabs panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
Binding affinity towards human ADORA1 (agonistic activity) in an in vitro assay with cellular components measured by scintillation counting
Assay data:3 Active, 227 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Binding affinity towards human ADORA1 in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:10 Active, 1 Activity ≤ 1 µM, 1182 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]-DPCPX from human recombinant adenosine A1 receptor at 10 uM after 60 mins by scintillation counting analysis relative to control
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of human alpha1A receptor at 1 uM relative to control
Binding affinity to adenosine A1 receptor (unknown origin) assessed as inhibition constant
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of Adenosine A1 receptor (unknown origin) at 10 uM
Binding affinity to human adenosine A1 receptor assessed as inhibition constant
Assay data:2 Tested
Inhibition of human CerS6
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed Citation
Inhibition of human CerS2
Inhibition of CerS6 (unknown origin) at 10 uM relative to control
SummaryPubMed Citation
Competitive inhibition of CerS2 in HPAC cells using DHSph as substrate by LC/MS/MS analysis
Inhibition of CerS2 in HPAC cells using DHSph as substrate
Displacement of [3H]cyclohexyladen from A1 adenosine receptor derived from rat cerebral cortical membrane assessed as inhibition constant
Assay data:2 Active, 2 Tested
Displacement of [3H]cyclohexyladen from A1 adenosine receptor derived from in guinea pig brain membrane assessed as inhibition constant
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to human adenosine A1 receptor assessed as dissociation constant
Antagonist activity at human A1 adenosine receptor
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Binding affinity to human A1 adenosine receptor assessed as inhibition constant
Assay data:3 Active, 1 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 3 Tested
Inhibition of human A1 adenosine receptor
Inhibition of human A1 adenosine receptor assessed as inhibition constant
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on