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Binding affinity to Trap1 (unknown origin) incubated for 24 hrs by fluorescence polarization assay
Assay data:5 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of TRAP1 NTD (unknown origin) by fluorescence polarization assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of TRAP1 (unknown origin)
Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to recombinant human TRAP1 assessed as inhibition constant incubated for 2 hrs by fluorescence polarization assay
Assay data:1 Tested
Inhibition of PU-FITC3 labeled Trap-1 (unknown origin) measured after 24 hrs by fluorescence polarization assay
Binding affinity to TRAP1 (unknown origin) by fluorescence polarization competitive binding assay
Assay data:4 Tested
Inhibition of TRAP1 in human HeLa cells assessed as reduction in SDHB protein expression at 25 uM after 12 hrs by Western blotting analysis
Assay data:4 Active, 4 Tested
Inhibition of PU-H71-FITC3 binding to recombinant full length TRAP1 (unknown origin) incubated for 2 hrs by fluorescence polarization assay
Assay data:30 Active, 26 Activity ≤ 1 µM, 31 Tested
Inhibition of FITC-GDA binding to human TRAP1 incubated for 2 hrs by fluorescence polarization assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
Assay data:4 Active, 2 Activity ≤ 1 µM, 14 Tested
Inhibition of TRAP1 in human PC3 cells assessed as increase in CHOP expression at 5 uM measured after 2 to 12 hrs by Western blot analysis
Assay data:1 Active, 2 Tested
Inhibition of TRAP1 in human PC3 cells assessed as reduction in SDHB expression at 5 uM measured after 2 to 12 hrs by Western blot analysis
Inhibition of TRAP1 in human PC3 cells assessed as reduction in SIRT3 expression at 5 uM measured after 2 to 12 hrs by Western blot analysis
Inhibition of TRAP1 in human PC3 cells assessed as increase in AMPK phosphorylation at 5 uM measured after 2 to 12 hrs by Western blot analysis
Inhibition of TRAP1 in human PC3 cells assessed as reduction in ATP concentration at 10 uM measured after 2 hrs
Inhibition of TRAP1 in human PC3 cells assessed as loss of mitochondrial membrane potential at 10 uM measured after 2 hrs by TMRM dye based flow cytometry
Assay data:2 Active, 2 Tested
Inhibition of TRAP1 in human PC3 cells assessed as increase in reactive oxygen species generation at 10 uM measured after 2 hrs by Mito-SOX probe based flow cytometry
Stimulation of recombinant wild-type human TRAP1 R114E/R402Q mutant ATPase activity expressed in Escherichia coli BL21 (DE3) up to 20 uM preincubated for 0.5 hrs followed by ATP addition and measured after 3 hrs by PiColorLock Gold reagent based colorimetric assay
Stimulation of recombinant wild-type human TRAP1 R402Q mutant ATPase activity expressed in Escherichia coli BL21 (DE3) up to 20 uM preincubated for 0.5 hrs followed by ATP addition and measured after 3 hrs by PiColorLock Gold reagent based colorimetric assay
Stimulation of recombinant wild-type human TRAP1 R114E mutant ATPase activity expressed in Escherichia coli BL21 (DE3) up to 20 uM preincubated for 0.5 hrs followed by ATP addition and measured after 3 hrs by PiColorLock Gold reagent based colorimetric assay
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