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Glutamate, Kainate Eurofins Panlabs panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
Binding affinity to GluK1 ligand binding domain (unknown origin)
SummaryPubMed CitationRelated BioAssays by Target
Binding affinity to GluK3 receptor (unknown origin)
Assay data:6 Active, 1 Activity ≤ 1 µM, 16 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to GluK2 receptor (unknown origin)
Assay data:4 Active, 1 Activity ≤ 1 µM, 15 Tested
Binding affinity to GluK1 receptor (unknown origin)
Assay data:4 Active, 16 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
KAINATE/R Eurofins SafetyScreen44 (BI)
Radioligand Binding Assay from US Patent US9656975: "Bicyclo[3.2.1]octyl amide derivatives and uses of same"
Assay data:10 Active, 1 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Glutamate, Non-Selective Eurofins-Panlabs radioligand binding assay
Glutamate, Kainate Eurofins-Panlabs radioligand binding assay
Assay data:5 Tested
Kainate CEREP ligand profiling
KAINATE/R Eurofins-Panlabs selectivity data (BI)
KAINATE/RA Cerep selectivity data (BI)
Negative allosteric modulation of rat GluK2 expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced current response at 30 uM at -40 mV holding potential in presence of concanavalin A by two-electrode voltage clamp method relative to glutamate alone
Assay data:1 Active, 2 Tested
Displacement of [3H]kainic acid from rat Glutamate receptor, ionotropic kainate at 10 uM after 60 mins by scintillation counting method relative to control
Assay data:2 Tested
Inhibition of rat brain Glutamate receptor, ionotropic kainate assessed as [3H]kainic acid uptake at 10 uM after 60 mins by scintillation counting analysis relative to control
Displacement of [3H]SYM2081 from recombinant homomeric rat GluK3 receptor expressed in baculovirus infected Sf9 insect cell membranes
Assay data:2 Active, 5 Tested
Displacement of [3H]SYM2081 from recombinant homomeric rat GluK2 receptor expressed in baculovirus infected Sf9 insect cell membranes
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