BioAssays for PubChem Compound (Select 42617993) - PubChem BioAssay - NCBI

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Select item 17989641.

CB Receptor Radioligand Binding Assay (Ki) from Article 10.1021/jm801534c: "Synthesis and evaluation of dibenzothiazepines: a novel class of selective cannabinoid-1 receptor inverse agonists."

Source:: BindingDB

Protein Targets:: Cannabinoid receptor 1; ...
Total:: 2

Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 11 Tested

AID:: 1798964

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 3499002.

Ratio of drug level in brain to plasma of ip dosed rat

Source:: ChEMBL

Assay data:2 Tested

AID:: 349900

Summary PubMed Citation

Select item 3496783.

Source:: ChEMBL

Assay data:2 Tested

AID:: 349678

Summary PubMed Citation

Select item 3496774.

Source:: ChEMBL

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 349677

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 3496765.

Clearance in rat

Source:: ChEMBL

Assay data:2 Tested

AID:: 349676

Summary PubMed Citation

Select item 3496756.

Half life in rat

Source:: ChEMBL

Assay data:2 Tested

AID:: 349675

Summary PubMed Citation

Select item 3496747.

Oral bioavailability in rat

Source:: ChEMBL

Assay data:2 Tested

AID:: 349674

Summary PubMed Citation

Select item 3496738.

Binding affinity to 5HTT

Source:: ChEMBL

Protein Target:: Sodium-dependent serotonin transporter

Assay data:3 Active, 3 Tested

AID:: 349673

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 3496729.

Binding affinity to DAT

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:3 Active, 3 Tested

AID:: 349672

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34967110.

Binding affinity to NET

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:3 Active, 3 Tested

AID:: 349671

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34967011.

Binding affinity to vasopressin 1A receptor

Source:: ChEMBL

Protein Target:: Vasopressin V1a receptor

Assay data:3 Active, 3 Tested

AID:: 349670

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966912.

Binding affinity to vasoactive intestinal peptide receptor

Source:: ChEMBL

Protein Target:: Vasoactive intestinal polypeptide receptor 1

Assay data:3 Active, 3 Tested

AID:: 349669

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966813.

Binding affinity to 5HT7 receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 7

Assay data:3 Active, 3 Tested

AID:: 349668

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966714.

Binding affinity to 5HT6 receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 6

Assay data:3 Active, 3 Tested

AID:: 349667

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966615.

Binding affinity to 5HT5A receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 5A

Assay data:3 Active, 3 Tested

AID:: 349666

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966516.

Binding affinity to 5HT4e receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 4

Assay data:3 Active, 3 Tested

AID:: 349665

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966417.

Binding affinity to 5HT3 receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 3A

Assay data:3 Active, 3 Tested

AID:: 349664

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966318.

Binding affinity to 5HT2B receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2B

Assay data:3 Active, 3 Tested

AID:: 349663

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966219.

Binding affinity to 5HT2A receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2A

Assay data:3 Active, 3 Tested

AID:: 349662

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966120.

Binding affinity to 5HT1B receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 1B

Assay data:3 Active, 3 Tested

AID:: 349661

Summary Compounds, Active PubMed Citation Related BioAssays by Target

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BioActivity

Active Compounds (58)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (2)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (4)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (4)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Literature Extraction (66)
BioAssays extracted from the literature

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