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Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB
Assay data:3598 Active, 421 Activity ≤ 1 nM, 2233 Activity ≤ 1 µM, 3598 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Inhibition of Escherichia coli AmpC assessed as nitrocefin hydrolysis by UV-Vis spectrophotometry
Assay data:1 Active, 1 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
qHTS Assay for Inhibitors of Tyrosyl-DNA Phosphodiesterase (TDP1)
Assay data:986 Active, 18 Activity ≤ 1 nM, 825 Activity ≤ 1 µM, 352260 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS Assay for Identification of Novel General Anesthetics
Assay data:256 Active, 6 Activity ≤ 1 nM, 1028 Activity ≤ 1 µM, 346372 Tested
qHTS for inhibitors of ROR gamma transcriptional activity
Assay data:16824 Active, 4 Activity ≤ 1 nM, 4465 Activity ≤ 1 µM, 309031 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS Assay for Inhibitors of RecQ-Like Dna Helicase 1 (RECQ1)
Assay data:1298 Active, 2 Activity ≤ 1 nM, 557 Activity ≤ 1 µM, 239513 Tested
VP16 counterscreen qHTS for inhibitors of ROR gamma transcriptional activity
Assay data:10662 Active, 5 Activity ≤ 1 nM, 1977 Activity ≤ 1 µM, 307648 Tested
qHTS Assay for Inhibitors of Bloom's syndrome helicase (BLM)
Assay data:697 Active, 70 Activity ≤ 1 nM, 398 Activity ≤ 1 µM, 354860 Tested
qHTS Assay for Inhibitors of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1)
Assay data:1227 Active, 548 Activity ≤ 1 nM, 13853 Activity ≤ 1 µM, 352185 Tested
qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen
Assay data:1950 Active, 291445 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia
Assay data:2061 Active, 409 Activity ≤ 1 µM, 291269 Tested
qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E)
Assay data:3597 Active, 395 Activity ≤ 1 µM, 229423 Tested
qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate
Assay data:16 Active, 90 Activity ≤ 1 µM, 236748 Tested
qHTS Assay for Inhibitors and Activators of Human alpha-Galactosidase From Spleen Homogenate
Assay data:19 Active, 89 Activity ≤ 1 µM, 239498 Tested
qHTS Assay for Inhibitors and Activators of N370S glucocerebrosidase as a Potential Chaperone Treatment of Gaucher Disease
Assay data:299 Active, 528 Activity ≤ 1 µM, 326770 Tested
qHTS Assay for Compounds that Induce Erasure of Genomic Imprints
Assay data:20 Active, 1 Activity ≤ 1 nM, 279 Activity ≤ 1 µM, 113755 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Quantitative High-Throughput Screen for Regulators of Epigenetic Control
Assay data:543 Active, 221 Activity ≤ 1 µM, 276569 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same Project
Experimentally measured binding affinity data derived from PDB
Assay data:3073 Active, 3073 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Texas Red Labeled MLL-derived Mutant Peptide
Assay data:615 Active, 1 Activity ≤ 1 nM, 686 Activity ≤ 1 µM, 266676 Tested
qHTS Assay for Inhibitors Targeting the Menin-MLL Interaction in MLL Related Leukemias: Competition With Fluorescein Labeled MLL-derived Peptide
Assay data:137 Activity ≤ 1 µM, 292510 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
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