BioAssays, Active for PubChem Compound (Select 16049170) - PubChem BioAssay - NCBI

Warning: The NCBI web site requires JavaScript to function. more...

Links from PubChem Compound

Items: 1 to 20 of 58

<< First< Prev

Page of 3

Select item 17989641.

CB Receptor Radioligand Binding Assay (Ki) from Article 10.1021/jm801534c: "Synthesis and evaluation of dibenzothiazepines: a novel class of selective cannabinoid-1 receptor inverse agonists."

Source:: BindingDB

Protein Targets:: Cannabinoid receptor 1; ...
Total:: 2

Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 11 Tested

AID:: 1798964

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 3496772.

Source:: ChEMBL

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 349677

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 3496103.

Displacement of [3H]SR141716 from human recombinant CB1 receptor expressed in HEK293 cells

Source:: ChEMBL

Protein Target:: Cannabinoid receptor 1

Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 15 Tested

AID:: 349610

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 3496094.

Inverse agonist activity at CB1 receptor assessed as repression of basal receptor activity by mammalian cell-based receptor selection and amplification technology method

Source:: ChEMBL

Protein Target:: Cannabinoid receptor 1

Assay data:19 Active, 19 Activity ≤ 1 µM, 20 Tested

AID:: 349609

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 3496735.

Binding affinity to 5HTT

Source:: ChEMBL

Protein Target:: Sodium-dependent serotonin transporter

Assay data:3 Active, 3 Tested

AID:: 349673

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 3496726.

Binding affinity to DAT

Source:: ChEMBL

Protein Target:: Sodium-dependent dopamine transporter

Assay data:3 Active, 3 Tested

AID:: 349672

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 3496717.

Binding affinity to NET

Source:: ChEMBL

Protein Target:: Sodium-dependent noradrenaline transporter

Assay data:3 Active, 3 Tested

AID:: 349671

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 3496708.

Binding affinity to vasopressin 1A receptor

Source:: ChEMBL

Protein Target:: Vasopressin V1a receptor

Assay data:3 Active, 3 Tested

AID:: 349670

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 3496699.

Binding affinity to vasoactive intestinal peptide receptor

Source:: ChEMBL

Protein Target:: Vasoactive intestinal polypeptide receptor 1

Assay data:3 Active, 3 Tested

AID:: 349669

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966810.

Binding affinity to 5HT7 receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 7

Assay data:3 Active, 3 Tested

AID:: 349668

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966711.

Binding affinity to 5HT6 receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 6

Assay data:3 Active, 3 Tested

AID:: 349667

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966612.

Binding affinity to 5HT5A receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 5A

Assay data:3 Active, 3 Tested

AID:: 349666

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966513.

Binding affinity to 5HT4e receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 4

Assay data:3 Active, 3 Tested

AID:: 349665

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966414.

Binding affinity to 5HT3 receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 3A

Assay data:3 Active, 3 Tested

AID:: 349664

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966315.

Binding affinity to 5HT2B receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2B

Assay data:3 Active, 3 Tested

AID:: 349663

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966216.

Binding affinity to 5HT2A receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 2A

Assay data:3 Active, 3 Tested

AID:: 349662

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966117.

Binding affinity to 5HT1B receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 1B

Assay data:3 Active, 3 Tested

AID:: 349661

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34966018.

Binding affinity to 5HT1A receptor

Source:: ChEMBL

Protein Target:: 5-hydroxytryptamine receptor 1A

Assay data:3 Active, 3 Tested

AID:: 349660

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34965919.

Binding affinity to thromboxane A2 receptor

Source:: ChEMBL

Protein Target:: Thromboxane A2 receptor

Assay data:3 Active, 3 Tested

AID:: 349659

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 34965820.

Binding affinity to ORL1 receptor

Source:: ChEMBL

Protein Target:: Nociceptin receptor

Assay data:3 Active, 3 Tested

AID:: 349658

Summary Compounds, Active PubMed Citation Related BioAssays by Target

<< First< Prev

Page of 3

Supplemental Content

Filters: Manage Filters

Refine your results

• What's this?

BioActivity

Active Compounds (58)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (2)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (4)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (4)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Literature Extraction (58)
BioAssays extracted from the literature

Actions on your results

View or Download BioAssay in PubChem

Find related data

Recent activity

Clear Turn Off Turn On

BioAssays, Active for PubChem Compound (Select 16049170) (58)
PubChem BioAssay

Your browsing activity is empty.

Activity recording is turned off.

Turn recording back on

See more...

You are here: NCBI > Chemicals & Bioassays > PubChem BioAssay