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CB Receptor Radioligand Binding Assay (Ki) from Article 10.1021/jm801534c: "Synthesis and evaluation of dibenzothiazepines: a novel class of selective cannabinoid-1 receptor inverse agonists."
Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Cmax in rat
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Displacement of [3H]SR141716 from human recombinant CB1 receptor expressed in HEK293 cells
Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 15 Tested
Inverse agonist activity at CB1 receptor assessed as repression of basal receptor activity by mammalian cell-based receptor selection and amplification technology method
Assay data:19 Active, 19 Activity ≤ 1 µM, 20 Tested
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