Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Cytotoxicity against human PC-3 cells assessed as inhibition of cell growth incubated for 48 hrs by MTT assay
Assay data:10 Active, 5 Activity ≤ 1 µM, 14 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Inhibition of N-terminal His10-StrepII tagged human ROCK2 catalytic domain (1 to 553 residues) expressed in Sf9 insect cells by HTRF assay
Assay data:49 Active, 81 Activity ≤ 1 µM, 90 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of FGFR-1 (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo kinase assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of GSK3beta (unknown origin) incubated for 20 mins in presence of 33P-ATP
Assay data:9 Active, 3 Activity ≤ 1 µM, 10 Tested
Inhibition of JNK1 (unknown origin) incubated for 20 mins in presence of 33P-ATP
Assay data:10 Active, 10 Activity ≤ 1 µM, 10 Tested
Inhibition of JNK2 (unknown origin) incubated for 20 mins in presence of 33P-ATP
Inhibition of human JNK2 incubated for 40 mins in presence of ATP and [gamma33P-ATP] by scintillation counting method
Assay data:10 Active, 10 Activity ≤ 1 µM, 11 Tested
Inhibition of human JNK1 incubated for 40 mins in presence of ATP and [gamma33P-ATP] by scintillation counting method
Assay data:10 Active, 9 Activity ≤ 1 µM, 11 Tested
Cytotoxicity against human NFF cells incubated for 72 hrs by resazurin staining based microplate reader assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 4 Tested
Inhibition of GST-tagged human full length LRRK2 transfected in HEK293T cells
Assay data:1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antiproliferative activity against human MDA-MB-468 cells assessed inhibition of cell growth incubated for 72 hrs by CCK-8 assay
Assay data:11 Active, 6 Activity ≤ 1 µM, 11 Tested
Inhibition of RSK1 (unknown origin)
Assay data:8 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 8 Tested
Inhibition of CDK6 (unknown origin) incubated for 60 mins in presence of ATP by luminescence based analysis
Assay data:16 Active, 14 Activity ≤ 1 µM, 16 Tested
Inhibition of GSK-3beta (unknown origin) expressed in Sf21 cells
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Binding affinity to SIK3 (unknown origin) transfected in HEK293 cells assessed as dissociation constant incubated for 1 hr by competitive binding assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity of AAK1 (unknown origin) assessed as dissociation constant
Assay data:17 Active, 2 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 17 Tested
Competitive inhibition of PKD3 (unknown origin) in presence of ATP
Competitive inhibition of PKD2 (unknown origin) in presence of ATP
Inhibition of PKD1 (unknown origin)
Assay data:15 Active, 3 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 16 Tested
Competitive inhibition of PKD1 (unknown origin) in presence of ATP
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on