BioAssays, activity concentration at/below 1 uM for PubChem Compound ( - PubChem BioAssay - NCBI

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Select item 19198001.

BRD9 Bromodomain TR-FRET Competition Binding Assay from US Patent US11773085: "Methods and compounds for treating disorders"

Source:: BindingDB

Protein Targets:: Bromodomain-containing protein 9; ...
Total:: 1

Assay data:67 Active, 84 Activity ≤ 1 µM, 84 Tested

AID:: 1919800

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147992.

Selectivity interaction (ITC) EUB0000205c BRPF3

Source:: ChEMBL

Protein Target:: Bromodomain and PHD finger-containing protein 3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914799

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147983.

Selectivity interaction (BromoScan panel) EUB0000205c BRPF3

Source:: ChEMBL

Protein Target:: Bromodomain and PHD finger-containing protein 3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914798

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147974.

Selectivity interaction (ITC) EUB0000205c BRPF1

Source:: ChEMBL

Protein Target:: Peregrin

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914797

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147965.

Selectivity interaction (BromoScan panel) EUB0000205c BRPF1

Source:: ChEMBL

Protein Target:: Peregrin

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914796

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147956.

Selectivity interaction (ITC) EUB0000205c BRD9

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 9

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914795

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147947.

Selectivity interaction (BromoScan panel) EUB0000205c BRD9

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 9

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914794

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147938.

Selectivity interaction (BromoScan panel) EUB0000205c BRD7

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 7

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914793

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19147919.

Selectivity interaction (ITC) EUB0000205c BRD1

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914791

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191479010.

Selectivity interaction (BromoScan panel) EUB0000205c BRD1

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914790

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191328511.

Affinity Biochemical interaction (AlphaScreen) EUB0000205c BRPF1

Source:: ChEMBL

Protein Target:: Peregrin

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913285

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191328412.

Affinity Biochemical interaction (AlphaScreen) EUB0000205c BRD1

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913284

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191299013.

Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000205c BRPF1

Source:: ChEMBL

Protein Target:: Peregrin

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1912990

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179486614.

Alpha Screen competitive assay from Article 10.1021/acschembio.7b00481: "Selective Targeting of Bromodomains of the Bromodomain-PHD Fingers Family Impairs Osteoclast Differentiation."

Source:: BindingDB

Protein Targets:: Bromodomain and PHD finger-containing protein 3; ...
Total:: 5

Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested

AID:: 1794866

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 166994715.

Alphascreen assay. Binding to BRPF1B (domain start/stop: M626-G740) by alphascreen assay

Source:: ChEMBL

Protein Target:: Peregrin

Assay data:7 Active, 4 Activity ≤ 1 µM, 7 Tested

AID:: 1669947

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 166993816.

Alphascreen assay. Binding to BRD1A (domain start/stop: E556-A688) by alphascreen assay

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 1

Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1669938

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 147576317.

Binding affinity to BRD9 (unknown origin) by isothermal titration calorimetry

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 9

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1475763

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 147576218.

Binding affinity to BRPF3 (unknown origin) by isothermal titration calorimetry

Source:: ChEMBL

Protein Target:: Bromodomain and PHD finger-containing protein 3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1475762

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 147575719.

Binding affinity to BRPF2 (unknown origin) by isothermal titration calorimetry

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1475757

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 147575220.

Binding affinity to BRPF1 (unknown origin) by isothermal titration calorimetry

Source:: ChEMBL

Protein Target:: Peregrin

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1475752

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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BioActivity

Active Compounds (38)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (1)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (38)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (38)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Literature Extraction (23)
BioAssays extracted from the literature
Other (15)
BioAssays deposited by other experimentalists

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